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Metabolism
Metabolism
♦PDE
(
0
)
Apremilast
Roflumilast
Sildenafil Citrate
Cilomilast
Tadalafil
Vardenafil HCl Trihydrate
Pimobendan
GSK256066
Deltarasin
Aminophylline
Icariin (Ieariline)
S- (+)-Rolipram
Rolipram
Anagrelide HCl
Dipyridamole
Cilostazol
Mardepodect (PF-2545920)
Dyphylline
Doxofylline
Milrinone
Irsogladine
Avanafil
Fenspiride HCl
Luteolin
Vardenafil
Mardepodect HCl (PF-2545920 HCl)
♦P450 (e.g. CYP)
(
0
)
Abiraterone
Abiraterone Acetate
Voriconazole
Avasimibe
Ketoconazole
Itraconazole
Fluconazole (UK49858)
Baicalein
Apigenin
Piperine
Diosmetin
Galeterone
Naringenin
Benzbromarone
Clarithromycin
Cobicistat (GS-9350)
PF-4981517
Ozagrel HCl
Ozagrel
TAK-700/Orteronel (s-isomer)
Pioglitazone HCl
Alizarin
Sodium Danshensu
Naringin
♦PPAR
(
0
)
Rosiglitazone maleate
Rosiglitazone
GW9662
T0070907
Pioglitazone
WY-14643 (Pirinixic Acid)
GSK3787
FH535
GW0742
Ciprofibrate
Fenofibrate
Gemfibrozil
Bezafibrate
Clofibric Acid
Rosiglitazone HCl
Troglitazone
♦Phospholipase
(
0
)
Varespladib (LY315920)
Clofazimine
Halobetasol Propionate
Polydatin
Tanshinone I (Tanshinone A)
Darapladib (SB-480848)
U73122
♦ DHFR
(
0
)
Methotrexate
Pralatrexate (racemic)
Pyrimethamine
Sulfameter
Pemetrexed Disodium Hydrate
♦Dehydrogenase
(
0
)
Mycophenolate Mofetil
Devimistat (CPI-613)
Leflunomide
AGI-5198
MK-8245
SW033291
NCT-501
Disulfiram
Trilostane
Vidofludimus
AGI-6780
PluriSIn-1 (NSC 14613)
Enoxolone
Ammonium Glycyrrhizinate
Gimeracil
Teriflunomide
Isovaleramide
Glycyrrhizin (Glycyrrhizic Acid)
Gossypol Acetate
♦ HSP
(
0
)
Tanespimycin (17-AAG)
Luminespib
17-DMAG (Alvespimycin) HCl
Ganetespib (STA-9090)
Elesclomol (STA-4783)
BIIB021
Onalespib (AT13387)
VER155008
KNK437
HSP990 (NVP-HSP990)
VER-50589
CH5138303
NMS-E973
VER-49009
XL888
SNX-2112 (PF-04928473)
KW-2478
PF-04929113 (SNX-5422)
Geldanamycin
NVP-BEP800
♦Carbonic Anhydrase
(
0
)
Dorzolamide HCl
Topiramate
U-104
Tioxolone
Methocarbamol
Brinzolamide
Dichlorphenamide
Methazolamide
Safinamide Mesylate
Rasagiline Mesylate
Tranylcypromine (2-PCPA) HCl
Moclobemide (Ro 111163)
Paeonol
Sennoside A
Safinamide
Tranylcypromine hemisulfate
♦MAO
(
0
)
♦FAAH
(
0
)
URB597
PF-3845
Biochanin A
JNJ-1661010
FAAH-IN-2
♦CETP
(
0
)
Anacetrapib (MK-0859)
Torcetrapib
Evacetrapib (LY2484595)
Dalcetrapib (JTT-705, RO4607381)
♦ Transferase
(
0
)
Tipifarnib
Lonafarnib
FK866 (APO866, Daporinad)
A922500
Tolcapone
LB42708
PF-04620110
FTI 277 HCl
♦HMG-CoA Reductase
(
0
)
Simvastatin
Rosuvastatin Calcium
Lovastatin
Fluvastatin Sodium
Atorvastatin Calcium
Pravastatin sodium
Clinofibrate
Mevastatin
Rosuvastatin
Rosuvastatin D3 Sodium
Rosuvastatin D6 Calcium
♦Hydroxylase
(
0
)
Nepicastat (SYN-117) HCl
Isotretinoin
Mildronate
Tetrahydropapaverine HCl
DMOG (dimethyloxaloylglycine)
(R)-Nepicastat HCl [RS-25560-198 HCl]
Telotristat Etiprate (LX 1606 Hippurate)
Telotristat (LP-778902)
♦IDO
(
0
)
NLG919
INCB024360 analogue
Indoximod (NLG-8189)
Epacadostat (INCB024360)
♦Retinoid Receptor
(
0
)
Tretinoin
Bexarotene (LGD-1069)
Adapalene
Tamibarotene
TTNPB (Arotinoid Acid)
♦Factor Xa
(
0
)
Rivaroxaban (BAY 59-7939)
Apixaban (BMS-56224701)
Edoxaban tosylate monohydrate (DU-176b)
Edoxaban
♦ AhR
(
0
)
StemRegenin 1 (SR1)
CH-223191
UM729
♦Ferroptosis
(
0
)
Erastin
Ferrostatin-1 (Fer-1)
Liproxstatin-1
♦Casein Kinase
(
0
)
Emodin
CX-4945 (Silmitasertib)
D 4476
Silmitasertib (CX-4945) Sodium
♦ NAMPT
(
0
)
Manidipine (CV-4093)
P7C3
GMX1778 (CHS828)
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