|
V75415
|
(S)-CVN424
|
1799968-74-3 |
(S)-CVN424 is a potent modulator of G protein-coupled receptor 6 (GPR6). |
|
V70305
|
2-Oleoylglycerol (2-octadecenoic acid monoglyceride; 2-glyceryl monooleate)
|
3443-84-3 |
2-Oleoylglycerol is a naturally occurring lipid in the diet. |
|
V77329
|
2-PCCA hydrochloride
|
|
2-PCCA HCl is a racemate and a GPR88 receptor agonist. |
|
V70558
|
[Ala17]-MCH
|
359784-84-2 |
[Ala17]-MCH is an analog of MCH and is a ligand for MCHR1 (Ki=0.16 nM) with greater selectivity for MCHR2 (Ki=34 nM). |
|
V70561
|
Ac-hMCH(6-16)-NH2
|
1053601-50-5 |
Ac-hMCH(6-16)-NH2 is a non-selective peptide agonist of MCH in human brain, with IC50s of 0.16 nM and 2.7 nM for MCH-1R and MCH-2R, respectively. |
|
V70556
|
AMG-076
|
1001438-96-5 |
AMG-076 is an orally bioactive, selective MCHR1 antagonist. |
|
V11653
|
AS1269574
|
330981-72-1 |
AS1269574 is a potent, orally bioactive GPR119 agonist with EC50 of 2.5 μM in HEK293 cells expressing human GPR119. |
|
V1806
|
AZD1981
|
802904-66-1 |
AZD1981 is a novel potent and selective CRTh2 (Chemoattractant receptor-homologous molecule expressed on TH2 cells; DP2-Prostaglandin D2 receptor 2, ) receptor antagonist with IC50 of 4 nM,it displayed>1000-fold selectivity over more than 340 other enzymes and receptors, including DP1. |
|
V86635
|
BI-9508
|
|
BI-9508 is a selective GPR88 agonist that crosses the blood-brain barrier. |
|
V75408
|
BigLEN(mouse)
|
501036-69-7 |
BigLEN(mouse) is a potent and specific agonist of orphan G protein-coupled receptor 171 (GPR171) with a Kd of approximately 0.5 nM. |
|
V75407
|
BigLEN(rat)
|
369377-66-2 |
BigLEN(rat) is a potent GPR171 agonist with EC50 of 1.6 nM. |
|
V78421
|
BigLEN(rat) TFA
|
|
BigLEN(rat) is a potent GPR171 agonist with EC50 of 1.6 nM. |
|
V75409
|
CID 2745687
|
264233-05-8 |
CID 2745687 is a specific, reversible and competitive GPR35 antagonist (inhibitor) with Ki of 12.8 nM. |
|
V75410
|
CID1231538
|
354126-20-8 |
CID1231538, a benzothiazole analog, is a potent GPR35 antagonist. |
|
V3995
|
CID1375606
|
313493-80-0 |
CID 1375606 is the first selective surrogate agonist of orphan G protein-coupled receptor (GPCR) GPR27 identified fromscreening a diversity-oriented synthesis library. |
|
V75416
|
CVN424
|
2254706-21-1 |
CVN424 is an orally bioactive and selective GPR6 inverse agonist/activator with a Ki of 9.4 nM and EC50 of 38 nM. |
|
V70557
|
Ethyl linolenate
|
1191-41-9 |
Ethyl linolenate is a fatty acid ethyl ester (FAEE). |
|
V70559
|
Ethyl linolenate-d5 (ethyl linolenate d5)
|
203633-16-3 |
Ethyl linolenate-d5 is the deuterated form of Ethyl linolenate. |
|
V75404
|
GPCR agonist-2
|
291528-35-3 |
GPCR agonist-2 (Compound 5j) is a GPCR GPR109b (HM74) agonist/activator with pEC50 of 6.51. |
|
V75405
|
GPR109 receptor agonist-2
|
957129-38-3 |
GPR109 receptor agonist (activator)-2 (Compound 5) is a selective GPR109a agonist with pEC50 of 5.53. |