Others 2

ADC Related

ADC Antibody ADC Cytotoxin ADC Linker ADCs Drug-Linker Conjugates for ADC
Angiogenesis

5-alpha Reductase ALK Bcr-Abl BTK EGFR FAK FLT3 HER-2 HIF Src Syk VDA VEGFR
Anti-infection

Antibiotic Arenavirus Bacterial CMV EBV Enterovirus Filovirus Fungal Gli HBV HCV HCV Protease HIV HSV Influenza Virus Parasite RABV Reverse Transcriptase RSV SARS-CoV TMV Virus Protease
Apoptosis

Apoptosis ASK Bcl-2 Caspase c-Myc c-RET Cytohesin DAPK Ferroptosis FKBP IAP Mdm2 p53 PD-1 PD-L1 PERK PKD Ras RIP kinase ROS Survivin Thymidylate Synthase TNF Receptor TNFa TRADD
Autophagy

Autophagy LRRK2 Mitophagy OGA ULK
Cell Cycle

Antifolate APC Aurora Kinase BMI-1 CDK Chk c-Myc Eukaryotic Initiation Factor G-quadruplex HDAC HSP Kinesin LIMK Mad2 Microtubule(Tubulin) Mps1 Nucleoside Antimetabolite/Analog Nur77 p21 PAK PERK PFKFB PLK PPAR Ras Rho ROCK SRPK TOPK Topoisomerase Wee1
Cytoskeletal Signaling

Arp2 3 Complex Bcr-Abl Cardiac Myosin Dynamin Gap Junction Protein HSP Integrin Kinesin Microtubule Associated MLCK Myosin PAK TACC3 Wntbeta-catenin
DNA Damage

ATM(ATR) CRISPR(Cas9) DNA alkylator DNA Stain DNA(RNA) Synthesis GAK HDAC HSP Nucleoside Antimetabolite(Analog) OGG1 p97 PARG PARP RAD51 RNR Sirtuin SMN Telomerase Topoisomerase
Endocrinology & Hormones

5-alpha Reductase ACE Adrenergic Receptor Androgen Receptor Aromatase Estrogenprogestogen Receptor Glucocorticoid Receptor GPR Mineralocorticoid Receptor RAAS THR TSH Receptor
Epigenetics

AMPK Aurora Kinase DNA Methyltransferase Epigenetic Reader Domain EZH1 2 HDAC HIF Histone Acetyltransferase Histone Demethylase Histone Methyltransferase JAK MAT MicroRNA MLL Pim PKC Protein Arginine Deiminase Sirtuin Small Interfering RNA (siRNA) SMYD

+MORE

Others 2

Others 2 related products

Cat No.	Product Name	CAS No.	Product Description
V3333	(S)-4CPG	134052-73-6	S)-4CPG [also known as (S)-4-Carboxyphenylglycine, and (S)-4C-PG] is a novel, potent,competitive and orally bioactive antagonist of metabotropic glutamate receptor 1 (mGluR) withselectivity for mGluR-1 over mGluR-5.
V3316	ARRY-797	1036404-17-7	ARRY-797 (also known as ARRY 371797) is a novel, potent and selective inhibitor of p38α (p38 mitogen-activated protein kinase).
V2975	B-Raf IN 1	950736-05-7	B-Raf IN 1 is a novel, potent and selective B-Raf inhibitor with IC50 of 24 nM; it is equally potent against c-Raf with IC50 of 25 nM.
V2989	BT-11	1912399-75-7	This product is discontinued due to commercial reason.
V3271	CB-1158 analog	1345810-21-0	CB-1158 analog (CB-1158, INCB01158 or Numidargistat analog) is a potent and orally bioavailable small-molecule inhibitor of the arginase with potential immunomodulating activities.
V3362	CP-55940 (CP 55,940)	83002-04-4	CP-55940 (CP-55,940;CP55,940) is a novel, potent and non-selective cannabinoid receptor agonist with Ki values of 0.58 and 0.69 nM for human recombinant CB1 and CB2, respectively.
V3177	FIPI HCl	1781834-93-2	FIPI HCl, the hydrochloride salt of FIPI which is formerly known as 5-Fluoro-2-indolyl deschlorohalopemide,is a derivative of halopemide which potently and selectively inhibits both PLD1 (phospholipase D) and PLD2 with IC50values of 25 nM and 20 nM, respectively.
V3197	GNF-6231	1243244-74-7	GNF-6231 is a novel, potent, orally active and selective Porcupine inhibitor that blocks Wnt signaling with IC50 of 0.8 nM (Wnt3a Co-culture RGA).
V3291	GSK-962	2049872-86-6	GSK-962 (also known as GSK962 or GSK962) is a negative control for GSK963 (also known as GSK963 or GSK963).
V3167	HDM201 R Enantiomer	1448867-42-2	HDM201 R Enantiomer is the R enantiomer of HDM201 (also called NVP-HDM201, HDM stands for human double minute 2 homolog).
V2911	HUHS015	1453097-13-6	HUHS015 is a novel and potent inhibitor of PCA-1/ALKBH3 (prostate cancer antigen-1/AlkB Homolog 3) both in vitro and in vivo that was discovered from the optimization of a hit compound identified during random screening using a recombinant PCA-1/ALKBH3.
V3040	JWH-133	259869-55-1	JWH-133 is a synthetic cannabinoid and a potent & selective agonist of the CB2 receptor with a Ki of 3.4nM and selectivity of ~ 200x for CB2 over CB1 receptors.
V3188	LGD-3303	917891-35-1	LGD-3303is a potent,selective, orally bioavailable, and non-sterdoidal androgen receptor modulator (SARM) with anabolic effects on muscle and cortical bone not observed with bisphosphonates.
V3259	Mavorixafor (AMD-070) triHCl	880549-30-4	MavorixafortriHCl (also known as AMD-1107, AMD070, X4P-001) is a potent, selective and orally bioavailable antagonist ofCXCR4 with anti-HIV activity.
V3328	MCOPPB 3HCl	1108147-88-1	MCOPPB 3HCl is a novel and potent nonpeptide agonist of nociceptin receptor with pKi of 10.07 and may be used as an anxiolytic agent.
V3220	ML239	1378872-36-6	ML239 was originally identified as a potent and selective inhibitor of breast cancer stem cells with an IC50of 1.16 μM, but recent studies (2016 Nature 12(2):109-16.
V3235	ML329	19992-50-8	ML329 is a potent small molecule inhibitor ofMITF (Micropthalmia-associated transcription factor) which inhibits TRPM-1 (melastatin, a MITF target gene) promoter activity with anIC50of 1.2 μM.
V3353	MRK-016 HCl	783331-24-8	MRK-016 HCl (MRK016; MRK 016) is a novel, potent, orally bioactive and selective negative allosteric modulator (inverse agonist) of α5 subunit-containing GABAA with nootropic properties.
V3275	NSC23005	6314-70-1	NSC23005 is a novel and potentp18inhibitor withED50of 5.21 nM in promoting Hematopoietic stem cells (HSCs) expansion in both murine and human models.
V3274	NSC23005 sodium	1796596-46-7	NSC23005 sodium is a novel and potentp18inhibitor withED50of 5.21 nM in promoting Hematopoietic stem cells (HSCs) expansion in both murine and human models.