5-HT receptors (Serotonin receptors) are a group of G protein-coupled receptors (GPCRs) and ligand-gated ion channels (LGICs) found in the central and peripheral nervous systems.5-HT1, 5-HT2, 5-HT3, 5-HT4, 5-HT5, 5-HT6, and 5-HT7 are the types. Both excitatory and inhibitory neurotransmission is mediated by them. The neurotransmitter serotonin, which serves as their inherently ligand, stimulates the serotonin receptors. Numerous neurotransmitters and hormones are released in response to stimulation of the serotonin receptors. Numerous biological and neurological functions, including aggression, anxiety, appetite, cognition, learning, memory, mood, nausea, sleep, and thermoregulation, are influenced by serotonin receptors. Many antidepressants, antipsychotics, anorectics, antiemetics, gastroprokinetic agents, antimigraine agents, hallucinogens, and entactogens are among the pharmaceuticals that target the serotonin receptors.
| Structure | Cat No. | Product Name | CAS No. | Product Description |
|---|---|---|---|---|
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V0999 | BRL-54443 | 57477-39-1 | BRL 54443 (BRL54443; BRL-54443) is a potent agonist of 5-HT1E and 5-HT1F receptor with important biological activity. |
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V2412 | BRL15572 free base | 734517-40-9 | BRL 15572 free base is an antagonist of 5-HT1D with around 60× selectivity over other related receptors. |
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V71230 | Bufotenidine | 487-91-2 | Bufotenidine is a naturally occurring alkaloid that works as a blocker of tryptophan receptors. |
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V0971 | Buspirone HCl (MJ90221) | 33386-08-2 | Buspirone HCl (MJ90221,MJ-90221,Buspar,MJ-9022-1, MJ9022 1, MJ9022-1), the hydrochloride salt of Buspirone which is anazapirone anolog,is a potent serotonergic 5HT1A receptor agonist with anti-psychotic effects. |
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V77632 | CART(62-76)(human,rat) TFA | CART(62-76)(human,rat) TFA is a neuropeptide (consisting of residues 62-76 of the CART peptide) that acts like a neurotransmitter. | |
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V85273 | CB2R/5-HT1AR agonist 1 | 2821085-76-9 | |
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V71138 | Cinitapride monotartrate | 1207859-16-2 | Cinitapride monotartrate is a 5-HT1A and 5-HT4 agonist. |
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V51787 | cis-(Z)-Flupentixol dihydrochloride | 51529-01-2 | DA D1/D2 receptor antagonist |
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V78797 | cis-Urocanic acid-13C3 ((Z)-Urocanic acid-13C3; cis-UCA-13C3) | cis-Urocanic acid-13C3 is a 13C (carbon 13)-labeled cis-Urocanic acid. | |
|
V11877 | Cisapride | 81098-60-4 | Cisapride (formerly R51619; R 51619; R-51619; Kaudalit; Prepulsid; Kinestase; Pridesia; Presid; Propulsid) is a benzamide-based nonselective agonist of serotonin 5-HT4 receptor. |
|
V7602 | Citalopram Hydrobromide (Lu 10-171) | 59729-32-7 | Citalopram Hydrobromide(Lu-10-171) is a potent and FDA approved antidepressant drug of the selective serotonin reuptake inhibitor (SSRI) class. |
|
V0990 | Clomipramine HCl (G34586) | 17321-77-6 | Clomipramine HCl (G-34586; G34586; Trade names: Anafranil, Clomicalm), the hydrochloride salt of clomipramine which is a tricyclic antidepressant (TCA), is a potent blocker of serotonin transporter (SERT), norepinephrine transporter (NET) dopamine transporter (DAT) with Ki of 0.14, 54 and 3 nM, respectively. |
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V0962 | Clozapine (HF 1854) | 5786-21-0 | Clozapine(LX 100129; HF1854, LX100129; Leponex; Fazaclo; CLOZARIL; Clozapin; Clozaril) is an atypical antipsychotic drug wand a 5-HT antagonist used in the treatment of schizophrenia. |
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V71142 | CP-135807 | 151272-90-1 | CP-135807 is an orally bioactive and selective 5-HT1D agonist (IC50=3.1 nM). |
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V4608 | CP-809101 HCl | 1215721-40-6 | CP-809101 HCl (CP809101), the hydrochloride salt ofCP-809101, is a novel, potent and selective 5-HT2C receptor agonist with antipsychotic effects. |
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V18922 | Cyamemazine | 3546-03-0 | Cyamemazine (Tercian; Cianatil; cyamepromazine) is a typical antipsychotic drug of the phenothiazine class. |
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V71222 | Cyamemazine-d6 | 1216608-24-0 | Cyamemazine-d6 is the deuterium labelled form of Cyamemazine. |
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V84822 | Cyanopindolol fumarate | 69906-86-1 | |
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V1918 | Cyclobenzaprine HCl (MK-130) | 6202-23-9 | Cyclobenzaprine HCl (also known as MK130; Flexeril), the hydrochloride salt of Cyclobenzaprine, is a potent muscle relaxant by blocking pain sensations, used as a medication for the treatment of skeletal muscle spasms and associated pain in acute musculoskeletal conditions. |
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V71209 | Cyclobenzaprine-d3 hydrochloride (MK130-d3 (hydrochloride)) | 1184983-42-3 | Cyclobenzaprine-d3 ( HCl) is the deuterium labelled form of Cyclobenzaprine HCl. |
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